Published March 24, 2016 | Version v1
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Shizukaol D, a Dimeric Sesquiterpene Isolated from Chloranthus serratus, Represses the Growth of Human Liver Cancer Cells by Modulating Wnt Signalling Pathway

  • 1. Fudan University
  • 2. Shanghai Jiaotong University
  • 3. University of Chicago

Description

Natural products have become sources of developing new drugs for the treatment of cancer. To seek candidate compounds that inhibit the growth of liver cancer, components of Chloranthus serratus were tested. Here, we report that shizukaol D, a dimeric sesquiterpene from Chloranthus serratus, exerted a growth inhibition effect on liver cancer cells in a dose- and time-dependent manner. We demonstrated that shizukaol D induced cells to undergo apoptosis. More importantly, shizukaol D attenuated Wnt signalling and reduced the expression of endogenous Wnt target genes, which resulted in decreased expression of β-catenin. Collectively, this study demonstrated that shizukaol D inhibited the growth of liver cancer cells by modulating Wnt pathway.

Data availability

All relevant data are within the paper and its Supporting Information files.

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Additional details

Identifiers

DOI
10.1371/journal.pone.0152012
Other
oai:uchicago.tind.io:7453

Funding

National Key Sci-Tech Special Project of China
2013ZX10002010
National Science Foundation of China
81301855

UChicago Information

Division(s)
Pritzker School of Medicine